Recent Highlights in the Discovery and Optimization of Crop Protection Products

Recent Highlights in the Discovery and Optimization of Crop Protections Products highlights the most prominent, recent results in the search for safe and effective new crop protection products. With a focus on the design, synthesis, optimization and/or structure-activity relationships of new chemistries targeting insect, disease, weed, nematode, vector and animal parasite control, the book also includes recent developments in crop enhancement chemistries and new approaches to crop protection products. The inclusion of information on testing tools, green chemistry approaches, and the latest discovery tools, like modeling, structure-based design, and testing tools makes this volume complete. Based on key presentations given at the 14th International IUPAC conference on Crop Protection, May 19-24, 2019 in Ghent, Belgium, this book includes the many exciting new discoveries and findings reported. It is designed to inspire additional research and advancement in the field. Based on science presented at the 2019 International Union of Pure and Applied Chemistry Conference on Crop ProtectionProvides real-world perspectives on pesticide and disease control progressPresents scientific developments from an international array of contributing authors INDICE: 1. Current trends and challenges in the Crop Protection2. New chemistries targeting insect control3. Discovery and optimization of a novel insecticide, broflanilide4. Studies on a novel insecticide, fluxametamide5. The discovery of Isocycloseram: A novel isoxazoline insecticide6. Discovery, synthesis and structure-activity relationship of tetraniliprole (VayegoTM), a novel diamide insecticide7. Cyclaniliprole: A novel diamide insecticide 8. Optimization of mesoionic pyrido[1,2-a] pyrimidinone insecticides & discovery of 3-biaryl analogs controlling lepidoptera species9. MNKE as a natural solution against insecticide-resistant pests10. Biology and Chemistry connected: The Development of Inscalis®11. Spiropidion discovery: road spectrum control of sucking pests and mites for multi-crop utility12. Synthesis and biological activity of a novel insecticide, benzpyrimoxan13. Design, synthesis and acaricidal activities of Cyflumetofen analogues based on carbon-silicon isosteric replacement14. Cycloclavine: A natural product with insecticidal potential. 15. Design, Synthesis of OfHex1 Inhibitors as Novel Pesticidal Leads.  16. New chemistries targeting disease control17. Discovery of ADEPIDYNTM.  18. Isoflucypram - A new succinate dehydrogenase inhibitor with unique structural features and performance.  19. Discovery of inpyrfluxam.  20. Isoflucypram - An innovative disease management tool with an unprecedented biological performance.  21. Chiral antifungal amides of 2-(2-oxazolinyl) aniline for the discovery of novel SDHIs.  22. Discovery of chiral antifungal ingredients with drimane as a new scaffold. 23. Discovery and biological profile of metyltetraprole 24. Discovery of florylpicoxamid, a new picolinamide for disease control  25. Revysol®: The new broad-spectrum fungicide of BASF SE 26. Synthesis and fungicidal activity of novel types of oxysterol-binding protein inhibitors. 27. Azole Carbinols as Fungicides28. Discovery of Pyruvate Kinase as a Fungicide Target by DARTS29. New chemistries targeting crop enhancement and animal parasite, nematode and vector control 30. Malaria Eradication, Agricultural Innovation and the ZERO by 40 Initiative31. Discovery and optimisation of novel compounds for the control of anopheline vectors of malaria32. Monoterpenoid esters as long-lasting spatial mosquito repellents33. Synergies between insecticide and parasiticide research: An evolving success story34. Antiparasitic dinitrile compounds for fly control in cattle35. Development of highly efficient plant virus disease prevention and control drug candidate NK0209 and NK033336. Discovery of novel antiviral agents based on marine natural products37. Design, synthesis and biological evaluation of Strigolactones derivatives for Crop Enhancement applications38. Use of synthetic plant defense elicitors as reduced-risk pesticide alternatives39. Discovery and optimization of 3(2H)-pyridazinone derivatives as novel plant activators40. CEDROZ®, new terpene nematicide against root knot nematode on Solanaceae and cucurbits41. Design, structural derivation and nematicidal activities of 1,2,3-Benzotriazin-4-one derivatives42. A novel class of priming agents with activity against fungi and nematodes43. Mulching efficacy and effect on soil microbial health of a sprayable, biodegradable polymeric mulch44. New chemistries targeting weed control 45. The discovery of aryl pyrrolidinone anilides: A new mode-of-action herbicide class that inhibits dihydroorotate dehydrogenase46. LuximoT herbicide - Rediscovering a dormant molecule47. Discovery and mode of action of cyclopyrimorate, a new paddy rice herbicide48. A new herbicide mode of action from a bioherbcicide component, spiceostatin c49. Resistance-gene directed discovery of a natural product herbicide with a new mode of action 50. Towards a Mechanistic Understanding of IGPD - A Potential Herbicide Target51. Isoxazolopyridines - A novel chemical cluster and a new mode of action for dicot weed control52. Discovery of New 4-Hydroxyphenylpyruvate Dioxygenase Inhibitors as Potential Herbicides53. TirexorTM - Design of a new resistance breaking PPO-inhibitor54. RinskorT active herbicide a new environmentally friendly tool for weed management in rice and aquatic environments55. Investigating c-h activation chemistry of n-phenyl azoles: discovery of a new class of herbicides56. Discovery of Novel Uracil herbicide by using Intermediate Derivatization Approach57. New approaches to crop protection products: discovery tools, green chemistry58. The use of green chemistry principles in the responsible design of crop protection processes and products59. Process route design of macrocyclic picolinamide fungicide X50760. New isothiazole inhibitors of protein biosynthesis: Towards the development of modern agchem products61. New approach to a bacterial causative crop disease and weed controls, using N-3-hydroxyoctanoyl-l- homoserine lactone, a tropolone biosynthetic activator for burkholderia plantarii62. COMPASS - A comprehensive model for pesticide activity in soils designed to guide the development and sustainable use of pesticides63. Nitrogen fertilization: A determining factor for efficiency of plant defense elicitors?64. Natural products: Most effective tool for creating green crop protection products65. Natural products: A source and inspiration for crop protection lead generation66. Photochromic insecticides for insect behavior modulation67. Exploring the molecular recognition properties of insect nicotinic acetylcholine receptors competitive modulators through multiscale molecular modeling68. A computational predictive approach for the discovery and optimization of new crop protection compounds 69. The agrochemical discovery portal: New computational platform for efficiently study pesticide and target interaction

• ISBN: 978-0-12-821035-2
• Editorial: Academic Press
• Encuadernacion: Rústica
• Páginas: 600
• Fecha Publicación: 31/01/2021
• Nº Volúmenes: 1
• Idioma: Inglés